Kinase Inhibitor [EPC]

42 drugs in this class with 1,444,234 total adverse event reports.

42 Drugs
1,444,234 Total Reports
750,312 Serious Reports
245,425 Death Reports
# Drug Name Generic Name Reports Serious Deaths
1 Tacrolimus TACROLIMUS 152,098 75,124 25,252
2 Tacrolimus Extended- TACROLIMUS EXTENDED-RELEASE CAPSULES 120,821 65,469 19,320
3 Pembrolizumab PEMBROLIZUMAB 100,428 73,843 18,175
4 Palbociclib PALBOCICLIB 94,183 46,263 10,456
5 Capecitabine CAPECITABINE 90,021 39,515 18,161
6 Ibrutinib IBRUTINIB 79,578 41,211 13,537
7 Ruxolitinib RUXOLITINIB 69,262 39,069 9,621
8 Letrozole LETROZOLE 60,074 28,867 5,933
9 Everolimus EVEROLIMUS 50,179 19,720 10,805
10 Dasatinib DASATINIB 36,591 13,929 3,681
11 Anastrozole ANASTROZOLE 35,755 12,218 2,401
12 Fulvestrant FULVESTRANT 32,192 17,023 4,876
13 Lenvatinib LENVATINIB 31,670 20,924 4,321
14 Osimertinib OSIMERTINIB 30,472 24,279 13,492
15 Octreotide OCTREOTIDE ACETATE 30,228 13,009 6,077
16 Ribociclib RIBOCICLIB 30,043 23,080 4,504
17 Nilotinib NILOTINIB 29,115 10,771 5,585
18 Pazopanib PAZOPANIB HYDROCHLORIDE 26,802 9,251 6,927
19 Trametinib TRAMETINIB 23,697 12,388 5,097
20 Exemestane EXEMESTANE 21,059 7,243 2,492
21 Hydroxyurea HYDROXYUREA 20,706 9,454 3,092
22 Dabrafenib DABRAFENIB 20,691 10,115 4,365
23 Sorafenib SORAFENIB 20,575 6,862 5,070
24 Axitinib AXITINIB 19,195 10,700 3,860
25 Abemaciclib ABEMACICLIB 18,718 13,866 1,388
26 Imatinib IMATINIB 17,162 9,026 3,043
27 Obinutuzumab OBINUTUZUMAB 15,802 8,904 2,119
28 Vigabatrin VIGABATRIN 14,291 4,502 1,370
29 Goserelin GOSERELIN 13,080 6,297 2,389
30 Sirolimus SIROLIMUS 12,953 6,993 2,096
31 Crizotinib CRIZOTINIB 12,556 5,423 3,761
32 Vemurafenib VEMURAFENIB 11,910 3,312 2,066
33 Basiliximab BASILIXIMAB 11,495 5,585 2,448
34 Acalabrutinib ACALABRUTINIB 11,444 10,195 2,493
35 Regorafenib REGORAFENIB 11,442 4,943 2,347
36 Avapritinib AVAPRITINIB 11,414 10,180 345
37 Entecavir ENTECAVIR 11,390 4,798 1,861
38 Erlotinib ERLOTINIB 9,597 5,214 4,329
39 Fam-Trastuzumab Deruxtecan-Nxki FAM-TRASTUZUMAB DERUXTECAN-NXKI 9,187 8,481 2,340
40 Gefitinib GEFITINIB 8,949 2,778 1,949
41 Bosutinib BOSUTINIB 8,855 4,196 764
42 Alpelisib ALPELISIB 8,554 5,292 1,217